Aspirin UPSA: litaelo tsa tšebeliso

Fomu ea tokollo

Matlapa a sebetsang hantle a bosoeu. Ha e qhibiliha ka metsing, ho ntšoa li-bubble tsa khase.

Motsoako o sebetsang: acetylsalicylic acid (500 mg), li-excipients: sodium carbonate anhydrous, anricrous ea sodium, anulinrous, sodium citrate anhydrous, sodium bicarbonate, crospovidone, aspartame, flavors ea tlhaho ea tlhaho, povidone.

Vitamin C: acetylsalicylic acid (330 mg), ascorbic acid (200 mg). Baeti: glycine, sodium benzoate, anhydrous citric acid, monosodium carbonate, polyvinylpyrrolidone.

Ho na le matlapa a 4 a sebetsang hantle moleng oa mochini oa foil oa aluminium o kentsoeng ka hare ka polyethylene. Marang-rang a 4 kapa a 25 hammoho le litaelo tsa tšebeliso ea pakete ea karete.

Vitamin C: Matlapa a 10 ka tube e le 'ngoe. Lerata le le leng kapa a mabeli ka lebokoseng la karete

Ketso ea pharmacological

E na le litlamorao tse khahlanong le ho ruruha, li-analgesic le antipyretic tse amanang le khatello ea cycloo oxygenase 1 le 2, e laolang mofuta oa li-prostaglandins. Fokotsa ho kopanya, ho khokhotheha ka liplatelete le thrombosis ka ho thibela ho kopana ha thromboxane A2 ka liplatelete, athe phello ea antiplatelet e phehella beke kamora ho nooa.

Monyetla oa sebopeho sa moriana o qhibilihang ha o bapisoa le asiti ea acetylsalicylic acid matlapeng ke ho monya ntho e sebetsang ka potlako le ka potlako.

Mofumahali

UPSA aspirin e kenngoa ka potlako ho feta aspirin e tloaelehileng. Palo e phahameng ea acetylsalicylic acid e fihlella ka metsotso e 20. Nako ea bophelo ba plasma e tsoa metsotso e 15 ho isa ho e 30. Acetylsalicylic acid e kenella ka har'a hydrolysis kahara plasma ka sebopeho sa salicylic acid. Salicylate e amahanngoa haholo le liprotheine tsa plasma. Mofuta oa moriana o hlaha ka pH ea moroto. Bophelo ba halofo ea acid e salicylic bo tsoa ho lihora tse 3 ho isa ho tse 9 mme o eketseha ka tekanyo e nkuoeng.

  • Bohloko bo bobebe kapa bo bobebe ho batho ba baholo ba mefuta e fapaneng: hlooho ea hlooho (ho kenyelletsa le e amanang le lefu la ho itlopa joala), leino le bohloko, migraine, neuralgia, radicular radicular syndrome, mesifa le bohloko bo kopaneng, bohloko nakong ea ho ea khoeling.
  • Keketseho ea mocheso oa 'mele mochesong le mafu a mang a tšoaetsanoang le a tšoaetsanoang (ho batho ba baholo le ho bana ba ka holimo ho lilemo tse 15).

Contraindication

  • Ho ruruha le ho ruruha ha lisele tsa mpa ea mpa ka mpeng, ho tsoa mali ka mpeng,
  • Portal hypertension,
  • "Aspirin" asthma,
  • Exorting Aortic Aneurysm,
  • Phenylketonuria,
  • Hemorrhagic diathesis, ho kenyelletsa hemophilia, telangiectasia, lefu la Willebrand, thrombocytopenia, hypoprothrombinemia, thrombocytopenic purpura,
  • Glucose-6-phosphate dehydrogenase e haelloang,
  • Hypersensitivity ho likarolo tsa Aspirin UPSA kapa litlhare tse ling tse seng khahlanong le ts'oaetso tsa steroidal,
  • Ho senya hampe le ho sebetsa ha meno,
  • Khaello ea Vitamin K

Setlhare se lumelloa ho nooa feela ho "trimester" ea bobeli ea bokhachane, ha e nooa nakong ea kemaro, ho khothaletsoa ho anyesa ho emisoa. Aspirin UPSA ha e sebelisoe ho bana ba ka tlase ho lilemo tse 15 ka lebaka la kotsi ea Reye syndrome.

Aspirin e lokela ho nkoa. ka tlhokomelo ka urate nephrolithiasis, hyperuricemia, pelo e emeng le ho peptic ulcer ea ka mpeng le duodenum ho anamnesis. Ha o sebelisa "aspirin", e lokela ho hopoloa hore e ka baka tlhaselo e matla ea gout e nang le bothata ba hona joale.

Tekanyetso le tsamaiso

Tekanyetso le kemiso ea ho amoheloa li khethoa ke ngaka e eang, hobane mona ntho e 'ngoe le e' ngoe e latela lilemo tsa mokuli.

Matlapa a sebetsang hantle a tlameha ho qhalwa pele ho 100-200 mg ea metsi a belisitsoeng ka mocheso oa kamore. Moriana o lokela ho nooa kamora lijo.

Ka bohloko bo boholo, o ka nka 400-800 mg ea acetylsalicylic acid makhetlo a 2-3 ka letsatsi (empa eseng ho feta 6 g ka letsatsi). Joaloka moemeli oa antiplatelet, ho sebelisoa litekanyetso tse nyane - 50, 75, 100, 300 kapa 325 mg ea ntho e sebetsang. Bakeng sa feberu, ho khothalletsoa ho nka 0.5-1 g ea acetylsalicylic acid ka letsatsi (haeba ho hlokahala, lethal dose le ka eketsoa ho 3 g).

Nako ea kalafo ha ea lokela ho feta matsatsi a 14.

Litla-morao

Ka tekanyetso e khothalletsoang, Aspirin UPSA hangata e mamelloa hantle. Khafetsa, ha u sebelisa lithethefatsi, ho ka hlaha mathata a latelang:

  • Letlalo la letlalo, "" aspirin triad ", bronchospasm le edincke's,
  • Mosebetsi o sa sebetseng oa renal,
  • Epistaxis, nako e eketsehang ea ho fetoha ha mali, marenene a tsoang mali,
  • Ho nyekeloa ke pelo, ho lahleheloa ke takatso ea lijo, ho hlatsa, ho tsoa mali ka mpeng, ho opeloa ke lets'ollo, lets'ollo,
  • Thrombocytopenia, leukopenia, anemia, hyperbilirubinemia.

Haeba litla-morao tse sa batleheng li hlaha, nka Aspirin UPSA e lokela ho emisoa.

Bongata

U lokela ho ba hlokolosi ka botaoa ba maqheku mme haholoholo baneng ba banyenyane (tšebeliso e feteletseng ea tahi kapa ho tahoa ka phoso, hangata e fumanoang baneng ba banyenyane), e ka lebisang lefung.

Matšoao a bokuli - ka tahi e lekanyelitsoeng, tinnitus e ka etsahala, tahlehelo ea litsebe, hlooho ea hlooho, ho tsekela, ho nyekeloa ke pelo ke sesupo sa bosholu. Lintho tsena li felisoa ka ho fokotsa tekanyetso. Ho tahoa haholo - hyperventilation, ketosis, alkalosis ea metabolism, komello, ho putlama ha pelo, ho se atlehe phefumong, hypoglycemia e phahameng.

Phekolo - ho tlosoa ha moriana kapele ka ho hlatsoa mpa. Ho kena sepetlele hang-hang setsing se ikhethang. Acid-base tekanyetso taolo. E qobelloang alkaline diuresis, hemodialysis, kapa peritoneal dialysis haeba ho hlokahala.

Ho sebelisana le lithethefatsi

Motsoako o nang le methotrexate o tiisitsoe, haholo litekanyetso tse phahameng (sena se eketsa chefo), ka li-anticoagulants tsa molomo ka tekanyetso e phahameng, kotsi ea ho tsoa mali e eketseha.

Motsoako o sa hlokahaleng - ka li-anticoagulants tsa molomo (ka tekanyetso e tlase, menyetla ea ho tsoa mali e eketseha), ka ticlopidine (e eketsa menyetla ea ho tsoa mali), ka li-uricosuric agents (ho fokotseha hoa ts'ebeliso ea uricosuric ho ka etsahala), le lithethefatsi tse ling tse thibelang mafu.

Motsoako o hlokang ts'ebetso ea ts'ireletso: le li-antidiabetesic agents (ka ho khetheha, sulfamide e fokotsang tsoekere) - phello ea hypoglycemic e eketseha, ka lithibela-mafu - nako le nako lipakeng tsa litekanyetso tsa li-antacid le lithethefatsi tsa salicylic li lokela ho bonoa (lihora tse 2), ka diuretics - tse nang le litekanyetso tse phahameng tsa lithethefatsi tsa salicylic, ho hlokahala hore ho boloka tekano e lekaneng metsi, lekola ts'ebetso ea renal qalong ea kalafo ka lebaka la ho hloleha ho matla ha methapo ea methapo ho mokuli ea nang le metsi, le li-corticoids (glucocorticoids) ) - le ka fokotseha salitsilemii nakong kalafo le corticoids le ho na kotsi ea ho e overdose ea salicylate mora qetello ea oona.

Bokhachane le pelehi

Setlhare sena se kopantsoe nakong ea bokhachane ho trimester ea I le III. Ka koteng ea bobeli ea kemolo, tekanyetso e le 'ngoe ea moriana o noang tekanyetso e ka ba teng feela ha molemo o lebelletsoeng ho mme o ka feta kotsi e ka bang teng ho lesea. Haeba ho hlokahala ho sebelisa moriana nakong ea lebone, ho anyesa ho lokela ho emisoe.

Litaelo tse khethehileng

Moriana o ka kenya letsoho ho tsoa mali, hammoho le ho eketsa nako ea ho ilela khoeli. Aspirin e eketsa kotsi ea ho tsoa mali haeba ho ka etsoa opereishene.

Ho bana, ha u fana ka moriana, ho bohlokoa ho nahana ka lilemo le boima ba 'mele.

Ka lijo tse se nang sodium ha li etsa lijo tsa letsatsi le letsatsi, ho lokela ho hopoloa hore tafole e 'ngoe le e' ngoe ea UPSA aspirin e nang le vithamine C e na le sodium e ka bang 485 mg.

Ho liphoofolo, phello ea teratogenic ea lithethefatsi e bonoa.

Matšoao a ho sebelisoa

Ho latela litaelo, Aspirin Oops e bontšoa bakeng sa:

  • Mafu a ho bata, a tšoaetsanoang le a tšoaetsanoang ho bana ba ka holimo ho lilemo tse 15 le batho ba baholo, a tsamaeang le feberu.
  • Bohloko bo bonolo kapa bo itekanetseng ho bakuli ba baholo ba mefuta e fapaneng: ho opeloa ke hlooho, ho kenyelletsa ho tahoa, migraine, leino, lefu la radicular syndrome, neuralgia, algomenorrhea, bohloko bo kopaneng le ba mesifa.

Tekanyetso le tsamaiso

Matlapa a Aspirin Oops pele a ts'ebeliso a lokela ho qhibiliha ka halofo ea khalase ea lero kapa metsi.

Bana ba kaholimo ho lilemo tse 15 le bakuli ba baholo ba beoa Letlapa le le leng ho fihlela makhetlo a 6 ka letsatsi. Ka bohloko bo boholo, mocheso o phahameng, tsamaiso ea nako e le 'ngoe ea Aspirin Ups e lumelloa ka tekanyetso ea matlapa a mabeli. Tekanyo e phahameng ea letsatsi le letsatsi ha ea lokela ho feta matlapa a 6 (3 g).

Bakuli ba tsofetseng Aspirin Ups ba fuoe Letlapa le le leng ho fihlela makhetlo a 4 ka letsatsi. Ho shebella khafetsa mokhoa oa ho sebelisoa ha Aspirin Oops ho u lumella ho fokotsa botebo ba syndrome ea bohloko le ho qoba ho eketseha ho eketsehileng ha mocheso oa 'mele.

Nako ea kalafo ea lithethefatsi ha ea lokela ho feta matsatsi a 5 ha e hlalosoa e le anesthetic le matsatsi a 3 e le antipyretic.

Ts'ebeliso ea moriana o noang litekanyetso tse phahameng ka nako e telele e ka baka matšoao a latelang a lithethefatsi tse ngata:

  • Hlooho e bohloko
  • Tsietsing
  • Ho utloa tahlehelo,
  • Matlafatso ea phefumoloho
  • Ho nyekeloa ke pelo, ho hlatsa,
  • Ho sitisoa ha pono
  • Khatello ea letsoalo
  • Ts'ebetso ea metabolism ea electrolyte,
  • Ho sitoa ho araba.

Haeba overdose e etsahala, mokuli o lokela ho hlatsa kapa a hlatsoe mpeng, a nke li-adsorbents le laxatives. Ho khothalletsoa ho ea sepetlele.

Litlamorao

Ts'ebeliso ea Aspirin Oops e ka baka litlamorao tse latelang:

  • Allergies: lekhopho la letlalo, bronchospasm, edema ea Quincke, "aspirin" triad (asthma ea bronchial, polyposis ea nko le sinuse sinuse, ho hloka mamello ho acetylsalicylic acid),
  • Sistimi ea urinary: ts'ebetso ea renal e senyehileng,
  • Mokhoa oa ho ja: ho nyekeloa ke pelo, ho hlatsa, lets'ollo, ho opeloa ke mpa, ho tsoa mali, ho eketsa ts'ebetso ea li-enzyme tsa sebete, ho fokotse takatso ea lijo,
  • Sisteme ea Hematopoietic: anemia, thrombocytopenia, hyperbilirubinemia, leukopenia,
  • Sistimi ea ho kopanya mali: hemorrhagic syndrome (ho tsoa mali, le maqhubu a mali), nako e eketsehang ea mali.

Mabakeng a ntlafatso ea litla-morao, mokuli o lokela ho khaotsa ho nka litlolo tsa mmele tsa Aspirin.

Aspirin UPSA

Litaelo tsa ho sebelisoa:

Aspirin UPSA ke setlhare se seng sa antiidalidal se sebelisang ho kokobetsa bohloko le ho fokotsa mocheso oa 'mele ho mafu a tšoaetsanoang kapa a tšoaetsanoang.

Lipehelo le maemo a polokelo

UPSA aspirin, ho latela litaelo, e lokela ho bolokoa ka moea o kenang hantle, moo bana ba ke keng ba e fumana le ho sirelletsoa sebakeng se omileng, se ommeng, ka mocheso o sa feteng 30 ° C.

Setlhare se fanoa ho tsoa litlolong tsa litlhare ntle le lengolo la ngaka, bophelo ba sona, se fumanehang ka litlhahiso tse kholo tsa moetsi, ke lilemo tse tharo. Kamora letsatsi la ho felloa ke nako, sehlahisoa se tlameha ho lahloa.

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Sebopeho sa moriana

Ntho e sebetsang e khethollang meaho ea lithethefatsi ke acetylsalicylic acid, dikahare ke 500 mg.

Lithako tse tlatselletsang tse khethollang sebopeho le thepa ea moemeli oa phekolo ke li-acric acid, metsoako ea sodium (carbonate le citrate), tatso le monko oa lamunu, aspartame, croslovidone, le likarolo tse ling.

Pholiso ea thepa

Aspirin matlapeng a draevecent e kenngoa ka potlako ho feta sehlahisoa se tšoanang, empa ka sebopeho sa eona se tloaelehileng. Khatello e phahameng ka ho fetisisa maling e thehoa metsotso e 1040 ka mor'a ho tsamaisoa. Sesebelisoa se sebetsang se hydrolyzed ho etsa salicylic acid, eo le eona e nang le phello ea kalafo. Likarolo tsena ka bobeli li hasana ka potlako ho pholletsa le 'mele, li hlola mokoallo oa placental, o kentsoeng lebese.

Acetylsalicylic acid e fetoloa ka har'a sebete, metabolites ea eona e tšeloa moroto.

Lokolla liforomo

Theko e tloaelehileng ke li-ruble tse 187.

Aspirin e hlahisoa ka mokhoa oa matlapa a atlehileng. Lipilisi ke sephara-cylindrical, li na le kotsi ea chamfer le e arohanang. Ha matlapa a felisoa, karabelo e ba teng ka ho lokolloa ha khabone.

Sehlahisoa se kenngoe ka marang-rang a lipilisi tse 4, ka har'a lipakete tsa karete - mela e mene, e tsamaeang le sengoloa.

Boimana le HB

Litokisetso tse nang le acetylsalicylic acid li ka se sebelisoe nakong tsena, haholo-holo ho basali ba 1st kapa 2nd trimester, ka lebaka la kotsi e kholo ea bokhachane ba methapo ea methapo ea methapo. Maemong a tlhokahalo e potlakileng, litekanyetso li lokela ho ba tse nyane ka hohle kamoo ho ka khonehang, mme kamohelo e lokela ho ba ea nakoana, e tšoaroe tlasa taolo le boikarabello ba ngaka.

Ka trimester ea 3, acid e hanyetsanoa ka tsela e ikhethang, kaha e ka kenya letsoho ho fetoleng boima ba masea, ho se sebetse hantle, ts'ebetso ea renal e sa sebetseng ho ngoana, ho fihlela kholong ea ho se lekane.

Ntle le moo, asiti e ka baka moferefere le ho tsoa mali ka nako e telele ho 'm'a kapa leseeng. Ho feta moo, litekanyetso tse nyane tsa aspirini le tsona lia li baka. Methapo e meholo ea asiti e sebelisoang qetellong ea bokhachane e lebisa ho holiseng mali. Masea a pele ho nako a tloaetse sena.

Basali ba nang le mongobo le bona ba tlameha ho lahla Aspirin Oops, hobane acetylsalicylic acid e khona ho kenella ka lebeseng.

Litlhokahalo tsa polokeho

Ka thupelo e telele ea Aspirin Oops, ho hlokahala hore ho etsoe liteko tsa mali le setofo, ho hlahloba boemo ba sebete.

  • Bakeng sa bakuli ba lefu la gout, lithethefatsi li ka baka ho eketseha, ka lebaka la bokhoni ba acetylsalicylic acid ho thibela tlhahiso ea methapo.
  • Bakuli ba ntseng ba buuoa ba khaotsa ho fokotsa ho tsoa mali nakong le kamora ho kenella.
  • Batho ba laolang ho kenella ha letsoai ba lokela ho hopola hore e teng ka sebopeho sa Aspirin Oops.

Tšebelisano ea lithethefatsi

Haeba ho na le tlhokahalo ea lithethefatsi tse ling, joale tsela ea Aspirin Ups e lokela ho etsoa ka hloko, hobane acetylsalicylic acid e kopana le likarolo tsa eona, e sotha thepa. Ka hona, ho hlokahala ho tsebisa ngaka ka lichelete tse nkuoeng.

  • Aspirin e ntlafatsa thepa ea antidiabetesic le anticonvulsants, diuretics.
  • Ha e kopantsoe le lithethefatsi tse nang le joala kapa joala, tšenyo ea mucous ea liprotheine tsa mokokotlo, matla le nako ea ho tsoa madi kahare lia matlafatsoa.
  • Aspirin e ke ke ea sebelisoa ka li-anticoagulants tsa molomo, ka lebaka la bofokoli ba phello ea morao le kotsi e eketsehileng ea ho tsoa mali. Haeba ho hlokahala, o hloka ho lekola khafetsa boemo ba mali bo kopanetsoeng.
  • Litokisetso tse nang le metsoako ea magnesium, aluminium, letsoai la calcium, li potlakisa ho tlosoa ha salicylates.

Litlamorao

Ho latela litekanyetso tse khothalletsoang ke baetsi kapa lingaka, litla-morao ha li hlahisoe, empa ha li khethoe:

  • Lipontšo tsa allergies - letlalo le phefumoloho (ho fihlela ho edema ea Quincke kapa bronchospasm)
  • Aspirin triad
  • Mathata a Stool, bohloko ba ka mpeng, ho tsoa mali ka hare, ho felloa ke takatso ea lijo
  • Tšenyo ea liphio
  • Ho tsoa mali, maqhubu a lutlang, nosetso le ho tsoa mali.

Haeba ho na le matšoao a belaetsang kamora ho nka Aspirin Oops, e tlameha ho hlakoloa ebe o etela ngaka.

Mefuta ea litekanyetso tsa Aspirin Oops

Indasteri ea meriana e hlahisa Aspirin Oops, e leng letlapa le lesoeu le bonojoana. Matlapa a na le 500 mg ea ntho e sebetsang - acetylsalicylic acid. Aspirin Oops e boetse e kenyelletsa bakuli. Tsena ke sodium carbonate, citric acid, sodium citrate. Sebopeho sa moriana o boetse o na le sodium bicarbonate, aspartame, flavors. Sephutheloana sena se na le matlapa a mane a sebetsang hantle a Aspirin Oops.

Matlapa a atlehileng a Aspirin Oops a na le 325 mg ea acetylsalicylic acid.

Tekanyetso le tsamaiso ea Aspirin Oops

Ho ea ka litaelo, Aspirin Oops e nkuoa ka molomo, 500-1000 mg ka letsatsi. Tekanyo e phahameng ea letsatsi le letsatsi ea Aspirin Oops e ka ba ligrama tse tharo. Ka tloaelo moriana o sebelisoa hanngoe kapa habeli ka letsatsi, o ka sebelisoa makhetlo a mararo. Pele o sebelisoa, letlapa la lithethefatsi le lokela ho qhibiliha ka khalase ea metsi. Haeba ho opeloa ke bohloko bo boholo mme ho na le mocheso o phahameng qalong ea lefu lena, joale o ka nka matlapa a mabeli hang-hang. Letsatsi ka lona u ke ke ua noa likoto tse fetang tse tšeletseng. Batho ba baholo ba laetsoe hore ba se ke ba nka litafole tse 'ne tsa Aspirin Oops. Joaloka antipyretic, Aspirin Oops e nkuoa matsatsi a mararo, joalo ka analgesic, o ka nka matsatsi a mahlano.

Bana ba ka tlase ho lilemo tse 'ne ha ba khothalletsoe ho fa Aspirin Oops. Ho tloha ho lilemo tse 4 ho isa ho tse 6 fana ka 200 mg ka letsatsi, lilemo tse 7-9 li nka 300 mg ka letsatsi. Bana ba kaholimo ho lilemo tse 12 ba ka nka 250 mg makhetlo a 2 ka letsatsi, ha tekanyetso ea letsatsi le letsatsi ha ea lokela ho ba ho feta 750 mg.

Ka infarction ea myocardial, bakuli ba ka nka Aspirin Oops ho tloha ho 40 ho isa ho 325 mg hang ka letsatsi. Setlhare se boetse se sebelisoa e le se thibelang ho kopana ha liplatelete. Tabeng ena, Aspirin Oops e nooa ka tekanyetso ea 325 mg ka letsatsi nako e telele.

Ho sebelisana le lithethefatsi tse ling

Ho latela litaelo, Aspirin Oops e ka ntlafatsa phello ea li-heparin le li-anticoagulants tsa molomo, hammoho le li-reserpine, lihormone tsa steroid. Setlhare se fokotsa litlamorao tsa lithethefatsi tse antihypertensive ha u ntse u li sebelisa. Ts'ebeliso ea Aspirin Oops le litlhare tse ling tse seng tsa steroid le tse thibelang mafu li ka hlahisa litlamorao tse mpe.

Lipehelo le maemo a polokelo

Sehlahisoa se loketse ts'ebeliso nakong ea lilemo tse 3 ho tloha ka letsatsi la tlhahiso. Bakeng sa ho qoba tahlehelo ea thepa ea kalafo, e lokela ho sireletsoa mochesong, khanya le mongobo o phahameng. Boloka ka mocheso ho fihlela ho 25 ° C, u be hole le bana.

Ho khetha sehlahisoa se nang le acetylsalicylic acid ha se bothata kajeno. Empa ka lebaka la likarolo tsa eona tsa bongaka, ho nkeloa sebaka hoa bongaka ho lokela ho etsoa ka thuso ea ngaka.

Bayer (Jeremane)

Karolelano ea karolelano: 258 r

Sehlahisoa se na le 400 mg ea ntho e sebetsang, e ruisitsoeng ka vithamine C (240 mg). Likarolo tse ling ke metsoako e bopehang sebopeho le solubility ea moriana. Setlhare se fumaneha ka mokhoa oa matlapa a maholo a masoeu ha a lokisa seno, ka lehlakoreng le leng ho na le leseli la "logo" la motho ea amehang ka tsela ea sefapano.

Moriana o nooa pilisi e le 'ngoe e qhibilihisitsoeng ka metsing, lethal dose le le leng le phahameng le lumeletsoeng ke matlapa a mabeli, e leng lethal dose la bobeli kamora lihora tse' ne.

Melemo:

  • Boleng bo botle
  • Ts'ebetso.

Mathata:

  • Ho ka etsahala hore a se ke a kula.

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