NEURORUBINE FORTE LACTAB N20

  • Matšoao a ho sebelisoa
  • Mokhoa oa kopo
  • Litlamorao
  • Ho sebelisana le lithethefatsi tse ling
  • Contraindication
  • Boimana
  • Bongata
  • Maemo a polokelo
  • Fomu ea tokollo
  • Sebopeho
  • Boikhethelo

Neurorubin-Forte Lactab - tokisetso ea motsoako o kopaneng o nang le li-vithamine tsa neurotropic tsa sehlopha B. Lisebelisoa tse sebetsang tsa lithethefatsi - livithamini B1, B6, B12 li ameha lits'ebetsong tsa biochemical tse netefatsang phetiso ea boipheliso haufi le methapo ea methapo, metabolism le metabolism ea babuelli ba methapo tsamaisong ea methapo.
Thiamine (vithamine B1), e hlophisitsoeng sebakeng sa lisele tsa methapo, e kenella ts'ebetsong ea tšusumetso ea methapo, e ntlafatsa ho nchafatsoa ha lisele tsa methapo. Ha ho thehoa likhahla tse kholo tsa thiamine maling, e khothalletsa nts'etsopele ea phello ea analgesic.
Pyridoxine (vithamine B6) e ama sebopeho le ts'ebetso ea lisele tsa methapo, pele ka ho laola metabolism ea amino acid, e thibelang ho bokelloa ha chefo ea neurotropic - ammonia. E nka karolo mohopolong oa baemeli ba fapaneng: catecholamines, histamine, GABA, e eketsa mabenkele a ikhethileng a magnesium, e phethang karolo ea bohlokoa ho metabolic, e leng, lits'ebetso tsa matla le tšebetso ea tsamaiso ea methapo.
Cyanocobalamin (vithamine B12) e baka metabolism ea nucleic acid mme e nka karolo, ka hona, ho boloka hematopoiesis, hape e fokotsa le neuroicic nociception.
Mofumahali
Thiamine mononitrate (vithamine B1) kamora hore tsamaiso ea molomo e khutsuoe ka duodenum le mala a manyane. Ka tekanyo e kholo, e kenngoa ka har'a sebete 'me metabolites ea eona e ka sehloohong ke thiaminocarboxylic acid le pyramine (2,5-dimethyl-4-aminopyridimine). Li-metabolites hammoho le palo e nyane ea thiamine e sa fetoloang li epolloa kahare le ka liphio.
Pyridoxine hydrochloride (vithamine B6) e kenella ka potlako ho tsoa mokokotlong oa mala. E na le metabolism ka har'a sebete ho boptjoa metabolites ea metabolic e sebetsang ea pyridoxalphosphate le pyridoxamine phosphate. Vitamin B6 e sebetsa e le coenzyme kamora phosphorylation ea sehlopha sa CH2OH maemong a 5, ka mantsoe a mang sebopeho sa pyridoxal 5-phosphate (PALP). Hoo e ka bang 80% ea PALP e kopana le liprotheine tsa plasma. Pyridoxine e bokellana ho isa tekanyong e kholo ea mesifa, sebete le tsamaiso ea methapo e bohareng. Litokisetso tsa ho qetela tsa metabolism ea pyridoxine ke 4-pyridoxyl acid, e ntlafalitsoeng ke liphio.
Cyanocobalamin (Vitamin B12). Sekhahla se ka sehloohong sa cyanocobalamin se ananeloa ka mor'a ho tlamaha Ntlo ea kahare ea Castle. Vitamin B12 e bokellana ho isa tekanyong e kholo ho sebete. T1 / 2 ho tsoa ho serum e ka ba matsatsi a 5, ho tloha sebete - e ka bang selemo se le seng. E pepisoa haholo ka bile le moroto.

Matšoao a ho sebelisoa

Neurorubin-Forte Lactab Ho khothalletsoa ho nka karolo ea kalafo e akaretsang:
- neuralgia, neuritis, polyneuritis,
- neuropathy, polyneuropathy (ho kenyeletsa lefu la tsoekere, joala),
- Lipontšo tsa Neurological tsa osteochondrosis ea lesapo la mokokotlo (sciatica, radiculopathy, mesnd-tonic syndromes).

Mokhoa oa kopo

Neurorubin-Forte Lactab khetha kahare, pele ho nako ea lijo. Lipilisi li entsoe ntle le ho hlafuna, li hlatsuoe ka metsi a lekaneng.
Batho ba baholo ba eletsoa hore ba noe lipilisi tse 1-2 /
Nako ea kalafo ke libeke tse 4. Monyetla oa ho etsa lithuto tse pheta-phetoang tsa kalafo o khethoa ke ngaka e ikhethileng.

Litlamorao

Litlamorao: ka linako tse ling - ho hlohlona, ​​hives, ho hema hanyane, edema ea Quincke, ho ts'oaroa ha anaphylactic.
Ho tsoa ts'ebetsong ea tšilo ea lijo: ka linako tse ling - ho nyekelwa ke pelo, ho tsoa mali ka mpeng, ho eketsa ts'ebetso ea AST.
Ho tsoa ho tsamaiso ea pelo: maemong a ikhethileng - tachycardia, ho oa, cyanosis, edema ea pulmonary.
Ba bang kaofela: nako le nako - ho fufuleloa ho sa lebelloang, ho ikutloa u se na thuso, ho tsekela, ho tšoenyeha, makhopho, ho sitisa secretion ea prolactin.

Ho sebelisana le lithethefatsi tse ling

Kaha pyridoxine hydrochloride e halefisa decarboxylation ea L-dopamine (levodopa) mme e ka fokotsa phello ea kalafo ea lithethefatsi ena kalafong ea bakuli ba nang le lefu la Parkinson, ts'ebeliso e tšoanang ea meriana ena ha ea lokela ho behelloa ka thoko.
Thiosemicarbazone le 5-fluorouracil li fokotsa katleho ea vithamine B1, ka hore ke bahanyetsi ba eona.
Li-antacids li liehisa ho amoheloa ha vithamine B1.

Fomu ea tokollo

Neurorubin-Forte Lactab - Lipilisi.
Ho paka - lipilisi tse 20.

Neurorubin-Forte Lactab e na le ntho e sebetsang: thiamine mononitrate (vit. B1) 200 mg, pyridoxine hydrochloride (vit. B6) 50 mg, cyanocobalamin (vit. B12) 1 mg.
Baeti: hypromellose, mannitol, cellulose e lerole, cellulose ea cellcrystalline, setlolo sa pregelatinized, magnesium stearate, colloidal silicon dioxide.
Sebopeho sa membrane ea filimi: hypromellose, macrogol 6000, talc, titanium dioxide (E171), erythrosine (E127).

NEURORUBINE forTE TABLETES N20
NEURORUBINE forTE TABLETES N20

Lebitso: Neurorubine

Ketso ea pharmacological:
Litokisetso tse rarahaneng tsa vithamine tse nang le livithamini tsa B tse tsamaisang metsi B. Li-vithamine tsa B li na le mefuta e mengata ea mesebetsi ea tlhaho, leha ho bile le litlamorao tse ts'oanang le tsa pharmacological, vithamine e 'ngoe le e' ngoe e na le phello e ikhethang 'meleng oa motho. Ka ho khetheha:
Vitamin B1 e nka karolo mafolofolo ho metabolism ea carbohydrate, ka ho haella ha eona keketseho ea palo ea li-lactic le pyruvic acid 'meleng e bonoa. E nka karolo ho deamination le transamination ea amino acid, ka hona ho laola metabolism ea protheine. Ho metabolism ea mafura, vithamine B1 e laola ho thehoa ha mafura a acid mme e thusa ho fetolela ha lik'habohaedreite hore ebe mafura. Mefuta e sebetsang ea vithamine ena e thusa ho matlafatsa sebopeho sa mala. Vitamin B1 e kenya tšebetsong mecha ea ion ka har'a metso ea methapo ea methapo, ka hona e ama ts'ebetso ea tšusumetso ho methapo ea methapo.

Vitamin B6 e kenya letsoho ho kopantsoeng ha li-enzyme, protheine le metabolism ea mafura. Sebopeho se mafolofolo sa vithamine ena se ameha liphethong tse fapaneng tsa enzymatic joalo ka coenzyme. Pyridoxine e laola motsoako oa li-neurotransmitters ka har'a methapo ea methapo e bohareng le e lipakeng, e nka karolo ho theheng membrane ea myelin ea neuron. E ntlafatsa tlhahiso ea matla, e nka karolo ho lipid le protheine ea metabolism, hape e laola synthet ea hemoglobin.

Vitamin B12 e bapala karolo ea bohlokoa ho metabolism ea protheine, e laola ho hlophisoa ha li-amino acid, li-purines le li-anemic acid. Cyanocobalamin e hlokahala bakeng sa mokhoa o tloaelehileng oa ts'ebetso ea myelination ea neuron le ho thehoa ha acetylcholine. Mekha e phahameng ea cyanocobalamin e thusa ho ntlafatseng litšusumetso tsa methapo le methapo ea methapo ea kutlo le ho hlohlelletsa nchafatso ea methapo ea methapo. O mong oa mesebetsi e ka sehloohong ea vithamine B12 ke phello ea eona ea antianemic. Cyanocobalamin e na le matla a hematopoietic, e hlohlelletsa erythropoiesis. Vithamine B12 e ntlafatsa hepatic hematopoiesis, e lokisa tsamaiso ea mali le ho thusa ho fokotsa cholesterol ea mali.

Neurorubin ea lithethefatsi e na le litekanyetso tse phahameng tsa kalafo ea li-vithamine tse kaholimo, tseo hammoho li kenya letsoho ho rarolleng mesebetsi ea tsamaiso ea methapo le ho laola lipid, carbohydrate le metabolism ea protheine. Ntle le moo, motsoako ona oa livithamini tsa B o thusa ho fokotsa bohloko le neuralgia ea limelo tse fapaneng.

Pharmacokinetics ea lithethefatsi Neurorubin e bakoa ke likarolo tsa pharmacokinetic tsa likarolo tsa eona tse teng:
Thiamine mononitrate ka mor'a ho tsamaisoa ka molomo, ho monngoa ha thiamine ho hlaha haholo ka mpeng e nyane, duodenum le jejunum. Karolo e nyane ea lithethefatsi e kenngoa ka har'a sebete, setlhare se kenngoa 'meleng ka ho etsoa hoa thiaminocarboxylic acid le pyramine. Metsotso e 30 ka mor'a ho buuoa ka molomo, ho kenella ha sethethefatsi maling ho tlase haholo ho feta litho le lisele. E ntšoa 'meleng ho tloha liponong le ka mala, e sa fetoheng le ka mokhoa oa metabolites.
Pyridoxine hydrochloride e kenelletse hantle ka mpeng, e thehiloe 'meleng ka sebopeho sa metabolites e sebetsang ea pyridoxal le pyridoxamine. Ntle le moo, pyridoxal-5-phosphate ke mofuta o sebetsang oa lithethefatsi, o phethang karolo ea coenzyme 'meleng. Pyridoxine e tšoauoa ka tekanyo e phahameng ea ho tlama liprotheine tsa plasma (ho fihla ho 80%). Cumulation ea lithethefatsi ka har'a sebete, mesifa le tsamaiso ea methapo e bohareng li ile tsa hlokomeloa. E tsoa 'meleng ke liphio ka mokhoa oa li-metabolites tse sebetsang le tse sa sebetseng.

Bakeng sa ho kenngoa ka mokhoa o tloaelehileng oa cyanocobalamin ka seterateng sa bona sa ka mpeng, ho ba teng ha ntlha ea Castle hoa hlokahala, ho netefatsang ho kenngoa ha lithethefatsi ka har'a potoloho ea systemic. Metabolism ea cyanocobalamin, ka lebaka la eona ho etsoa ha adenosylcobalamin metabolite, e hlaha liseleng. E tšeloa ka har'a moroto le bile. E bokellana sebeteng. Bophelo ba halofo ea lithethefatsi ho tsoa ho lero la mali ke matsatsi a 5, ho tloha liseleng tsa sebete - nako e ka bang selemo.


Matšoao a sebeliso:
Setlhare sena se sebelisoa maemong a tsamaeang le matšoao a hypovitaminosis ea livithamini tsa sehlopha B 'meleng.
Matlapa a koahetsoeng ka filimi, Neurorubin-Forte Lactab a sebelisoa kalafong e rarahaneng ea maloetse a joalo:
Bohloko ba mefuta e sa foleng le e sa foleng ea neuritis le polyneuritis,
Neuralgia, le tšenyo ea methapo ea methapo nakong ea botaoa le lintho tse fapaneng, ho kenyeletsa tahi le tahi ea lithethefatsi,
Lefu la tsoekere la polyneuropathy.
Tharollo ea ente Neurorubin e sebelisoa e le monotherapy kapa hammoho le lithethefatsi tse ling bakeng sa mafu a joalo:
Li-neuropathies, ho kenyeletsa le peripheral, tse bakoang ke joala.
Diabetes polyneuropathies.
Vitamin B hypovitaminosis, beriberi e omeletseng le e metsi.
Neuralgia, ho kenyelletsa cervicobrachial le trigeminal neuralgia.
Anuritis e sa foleng le e sa foleng le polyneuritis ea li-etiologies tse fapaneng.


Mokhoa oa ts'ebeliso:
Melemo ea lithethefatsi le nako ea kalafo e khethoa ke ngaka e etsoang ka bomong bakeng sa mokuli ka mong.
Matlapa a koahetsoeng ka filimi, Neurorubin-Forte Lactab a nooa ka molomo ka metsi a lekaneng, haholo pele ho lijo kapa nakong ea lijo, ha ho khothalletsoe ho arola kapa ho hlafuna matlapa a koahetsoeng ka filimi. Hangata batho ba baholo ba fuoa matlapa a 1-2 ka letsatsi. Nako ea kalafo hangata hangata e le 1 khoeli.

Tharollo ea ente Neurorubin e sebelisoa bakeng sa ente ea methapo ea kutlo; liente li khothaletsoa sethaleng se kaholimo sa mesifa ea gluteal.
Litekanyetso tsa lithethefatsi le khafetsa ea liente li latela botebo ba hypovitaminosis.
Maemong a matla, 3 ml ea lithethefatsi hangata e tsamaisoa letsatsi le leng le le leng kapa ka nako e le ngoe ka matsatsi a 2 ho fihlela tekanyo ea methapo ea bohloko e fokotseha, kamora moo ba fetohelang 3 ml ea moriana makhetlo a 1-2 ka matsatsi a 7.
Maemong a boima bo leka-lekaneng, 3 ml ea lithethefatsi hangata e tsamaisoa makhetlo a 1-2 ka matsatsi a 7.
Nako ea phekolo ea botsoali le Neurorubin e itšetlehile ka sesosa sa hypovitaminosis. Ha u etsa kalafo ea lithethefatsi ea nako e telele, li-paramente tsa laboratori li lokela ho betoa leihlo likhoeli tse ling le tse ling tse 6.


Litlamorao:
Ha o sebelisa lithethefatsi ho bakuli, ho ile ha hlokomeloa litlamorao tse latelang:
Ho tsoa ho tsamaiso ea tšilo ea lijo: ho nyekeloa ke pelo, ho hlatsa, ho eketseha ha lipilisi tsa hepatic maling. Ho bakuli ba nang le kutloisiso e eketsehileng ea motho ka mong, ho tsoa mali ho ile ha hlokomeleha ha ho nooa moriana.
Ho tloha tsamaisong ea methapo ea methapo e bohareng le e poteletseng: bofokoli, hlooho ea hlooho, ho tsekela. Maemong a ikhethileng, ho tšoenyeha, ho teneha ho eketsehileng le ho tšoenyeha ho ile ha hlokomeloa. Ha ba sebelisa lithethefatsi ka tekanyetso e phahameng, bakuli ba bang ba hlokometse ketsahalo ea "peripheral sensory neuropathy" e hlahang kamora ho khaotsa lithethefatsi.

Ho tsoa ho tsamaiso ea pelo: tachycardia, ho putlama ha mali (ho bonoang feela ho bakuli ba nang le kutloisiso e eketsehileng ea motho ka mong).
Mekhoa ea ho kulisa: ho hlohlona ha letlalo, lekhopho, urticaria, ha u sebelisa litekanyetso tse phahameng tsa moriana ho bakuli, nts'etsopele ea makhopho e ile ea lemohuoa.
Litla-morao tse ling: cyanosis, edema ea pulmonary, mofufutso. Ho bakuli ba nang le hypersensitivity ho likarolo tsa moriana, ho ka hlaha maikutlo a anaphylactoid, ho kenyeletsa edema ea Quincke. Ka tsamaiso ea batsoali ea lithethefatsi ho bakuli ba nang le hypersensitivity ho livithamini tsa B, ho ka ba le tšohanyetso ea tšohanyetso.


Contraindication:
Ho eketsa kutloisiso ea motho ka mong likarolo tsa moriana.
E laetsoe ka hloko ho bakuli ba nang le psoriasis, hobane cyanocobalamin e ka tsosa ho senyeha ho psoriasis.
Neurorubin ea lithethefatsi ka mokhoa oa tharollo ea ente ha e sebelisoe nakong ea bokhachane le pelehi, hammoho le kalafo ea bana ba ka tlase ho lilemo tse 16.


Boimana
Setlhare se tšela mekoallo ea hematoplacental 'me se ikemiselitse ho lebese la matsoele. Ha ho na datha mabapi le polokeho ea moriana nakong ea kemolo le ho lactation. Lithethefatsi nakong ea kemolo li ka laeloa ke ngaka e tlang haeba phaello e lebelletsoeng ho mme e feta kotsi e ka bang teng ho lesea. Haeba ho hlokahala ho fana ka moriana nakong ea lebone, hoa hlokahala ho etsa qeto ea ho khaotsa ho anyesa.


Ho sebelisana le lithethefatsi tse ling:
Ka tšebeliso e le 'ngoe, sethethefatsi sena se fokotsa phello ea kalafo ea levodopa, e lokelang ho tsotelloa ha u phekola bakuli ba nang le lefu la Parkinson le ho qoba tšebeliso e tšoanang ea meriana ena.
Ka tšebeliso e tšoanang, Neurorubin ea lithethefatsi e ntlafatsa chefo ea isoniazid.
Neurorubin ka lebaka la vithamine ea eona ea B6 e khona ho fokotsa katleho ea altretamine ka tšebeliso e tšoanang.
Thiosemicarbazone le fluorouracil ke bahanyetsi ba vithamine B1.
Lithethefatsi tse nang le envelop le thepa ea antacid li fokotsa ho amoheloa ha lithethefatsi Neurorubin-Forte Lactab.


Bongata
Ka tšebeliso ea lithethefatsi tse ngata ho bakuli, keketseho ea ho teba ha litlamorao e bonoa.
Ha ho na litlhare tse tobileng. Haeba ho na le overdose, gastric lavage le tsamaiso ea li-enterosorbents li bontšoa. Phekolo ke letšoao. Ka nts'etsopele ea anaphylactic makala, li-glucocorticosteroids bakeng sa ts'ebeliso ea systemic le li-antihistamines li sebelisoa.


Foromo ea tokollo:
Litafole, koaetsoe ka filimi, likotoana tse 10 ka blister, 2 lithutsoana ka lebokoseng la karete.
Tharollo ea ente ea 3 ml ka ampoule, ampoules tse 5 ka lebokoseng la karete.


Maemo a polokelo:
Setlhare se khothalletsoa hore se bolokoe sebakeng se omileng hole le khanya ea letsatsi. Matlapa a Neurorubin-Forte Lactab a khothalletsoa hore a bolokoe ka mocheso oa likhato tse 15 ho isa ho 25 tsa Celsius.
Tharollo ea ente Neurorubin e khothalletsoa hore e bolokoe ka mocheso oa likhato tse 2 ho isa ho tse 8 tsa Celsius.
Bophelo ba sehatsetsing sa moriana ka mokhoa oa tharollo ea ente ke lilemo tse 3.
Bophelo ba sehatsetsing ba lithethefatsi ka mokhoa oa matlapa ke lilemo tse 4.


Synonyms:
Neurovitan, Milgamma.


Moetso:
3 ml (1 ampoule) ea ente e na:
Thiamine hydrochloride - 100 mg,
Pyridoxine hydrochloride - 100 mg,
Cyanocobalamin - 1 mg.
Bahlomphehi.

Letlapa le 1 le koahetsoeng ka filimi le na le:
Thiamine mononitrate - 200 mg,
Pyridoxine hydrochloride - 50 mg,
Cyanocobalamin - 1 mg.
Bahlomphehi.


Hlokomela!
Pele o sebelisa lithethefatsi Neurorubin o lokela ho bona ngaka. Buka ena e fanoa phetolelong ea mahala ebile e etselitsoe merero ea tlhahisoleseling feela. Bakeng sa tlhaiso-leseling e batsi, ka kopo sheba litlhaloso tsa moetsi.
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Lebitso: Neurorubine

Ketso ea pharmacological:
Litokisetso tse rarahaneng tsa vithamine tse nang le livithamini tsa B tse tsamaisang metsi B. Li-vithamine tsa B li na le mefuta e mengata ea mesebetsi ea tlhaho, leha ho bile le litlamorao tse ts'oanang le tsa pharmacological, vithamine e 'ngoe le e' ngoe e na le phello e ikhethang 'meleng oa motho. Ka ho khetheha:
Vitamin B1 e nka karolo mafolofolo ho metabolism ea carbohydrate, ka ho haella ha eona keketseho ea palo ea li-lactic le pyruvic acid 'meleng e bonoa. E nka karolo ho deamination le transamination ea amino acid, ka hona ho laola metabolism ea protheine. Ho metabolism ea mafura, vithamine B1 e laola ho thehoa ha mafura a acid mme e thusa ho fetolela ha lik'habohaedreite hore ebe mafura. Mefuta e sebetsang ea vithamine ena e thusa ho matlafatsa sebopeho sa mala. Vitamin B1 e kenya tšebetsong mecha ea ion ka har'a metso ea methapo ea methapo, ka hona e ama ts'ebetso ea tšusumetso ho methapo ea methapo.

Vitamin B6 e kenya letsoho ho kopantsoeng ha li-enzyme, protheine le metabolism ea mafura. Sebopeho se mafolofolo sa vithamine ena se ameha liphethong tse fapaneng tsa enzymatic joalo ka coenzyme. Pyridoxine e laola motsoako oa li-neurotransmitters ka har'a methapo ea methapo e bohareng le e lipakeng, e nka karolo ho theheng membrane ea myelin ea neuron. E ntlafatsa tlhahiso ea matla, e nka karolo ho lipid le protheine ea metabolism, hape e laola synthet ea hemoglobin.

Vitamin B12 e bapala karolo ea bohlokoa ho metabolism ea protheine, e laola ho hlophisoa ha li-amino acid, li-purines le li-anemic acid. Cyanocobalamin e hlokahala bakeng sa mokhoa o tloaelehileng oa ts'ebetso ea myelination ea neuron le ho thehoa ha acetylcholine. Mekha e phahameng ea cyanocobalamin e thusa ho ntlafatseng litšusumetso tsa methapo le methapo ea methapo ea kutlo le ho hlohlelletsa nchafatso ea methapo ea methapo. O mong oa mesebetsi e ka sehloohong ea vithamine B12 ke phello ea eona ea antianemic. Cyanocobalamin e na le matla a hematopoietic, e hlohlelletsa erythropoiesis. Vithamine B12 e ntlafatsa hepatic hematopoiesis, e lokisa tsamaiso ea mali le ho thusa ho fokotsa cholesterol ea mali.

Neurorubin ea lithethefatsi e na le litekanyetso tse phahameng tsa kalafo ea li-vithamine tse kaholimo, tseo hammoho li kenya letsoho ho rarolleng mesebetsi ea tsamaiso ea methapo le ho laola lipid, carbohydrate le metabolism ea protheine. Ntle le moo, motsoako ona oa livithamini tsa B o thusa ho fokotsa bohloko le neuralgia ea limelo tse fapaneng.

Pharmacokinetics ea lithethefatsi Neurorubin e bakoa ke likarolo tsa pharmacokinetic tsa likarolo tsa eona tse teng:
Thiamine mononitrate ka mor'a ho tsamaisoa ka molomo, ho monngoa ha thiamine ho hlaha haholo ka mpeng e nyane, duodenum le jejunum. Karolo e nyane ea lithethefatsi e kenngoa ka har'a sebete, setlhare se kenngoa 'meleng ka ho etsoa hoa thiaminocarboxylic acid le pyramine. Metsotso e 30 ka mor'a ho buuoa ka molomo, ho kenella ha sethethefatsi maling ho tlase haholo ho feta litho le lisele. E ntšoa 'meleng ho tloha liponong le ka mala, e sa fetoheng le ka mokhoa oa metabolites.
Pyridoxine hydrochloride e kenelletse hantle ka mpeng, e thehiloe 'meleng ka sebopeho sa metabolites e sebetsang ea pyridoxal le pyridoxamine. Ntle le moo, pyridoxal-5-phosphate ke mofuta o sebetsang oa lithethefatsi, o phethang karolo ea coenzyme 'meleng. Pyridoxine e tšoauoa ka tekanyo e phahameng ea ho tlama liprotheine tsa plasma (ho fihla ho 80%). Cumulation ea lithethefatsi ka har'a sebete, mesifa le tsamaiso ea methapo e bohareng li ile tsa hlokomeloa. E tsoa 'meleng ke liphio ka mokhoa oa li-metabolites tse sebetsang le tse sa sebetseng.

Bakeng sa ho kenngoa ka mokhoa o tloaelehileng oa cyanocobalamin ka seterateng sa bona sa ka mpeng, ho ba teng ha ntlha ea Castle hoa hlokahala, ho netefatsang ho kenngoa ha lithethefatsi ka har'a potoloho ea systemic. Metabolism ea cyanocobalamin, ka lebaka la eona ho etsoa ha adenosylcobalamin metabolite, e hlaha liseleng. E tšeloa ka har'a moroto le bile. E bokellana sebeteng. Bophelo ba halofo ea lithethefatsi ho tsoa ho lero la mali ke matsatsi a 5, ho tloha liseleng tsa sebete - nako e ka bang selemo.

Matšoao a sebeliso:
Setlhare sena se sebelisoa maemong a tsamaeang le matšoao a hypovitaminosis ea livithamini tsa sehlopha B 'meleng.
Matlapa a koahetsoeng ka filimi, Neurorubin-Forte Lactab a sebelisoa kalafong e rarahaneng ea maloetse a joalo:
Bohloko ba mefuta e sa foleng le e sa foleng ea neuritis le polyneuritis,
Neuralgia, le tšenyo ea methapo ea methapo nakong ea botaoa le lintho tse fapaneng, ho kenyeletsa tahi le tahi ea lithethefatsi,
Lefu la tsoekere la polyneuropathy.
Tharollo ea ente Neurorubin e sebelisoa e le monotherapy kapa hammoho le lithethefatsi tse ling bakeng sa mafu a joalo:
Li-neuropathies, ho kenyeletsa le peripheral, tse bakoang ke joala.
Diabetes polyneuropathies.
Vitamin B hypovitaminosis, beriberi e omeletseng le e metsi.
Neuralgia, ho kenyelletsa cervicobrachial le trigeminal neuralgia.
Anuritis e sa foleng le e sa foleng le polyneuritis ea li-etiologies tse fapaneng.

Mokhoa oa ts'ebeliso:
Melemo ea lithethefatsi le nako ea kalafo e khethoa ke ngaka e etsoang ka bomong bakeng sa mokuli ka mong.
Matlapa a koahetsoeng ka filimi, Neurorubin-Forte Lactab a nooa ka molomo ka metsi a lekaneng, haholo pele ho lijo kapa nakong ea lijo, ha ho khothalletsoe ho arola kapa ho hlafuna matlapa a koahetsoeng ka filimi. Hangata batho ba baholo ba fuoa matlapa a 1-2 ka letsatsi. Nako ea kalafo hangata hangata e le 1 khoeli.

Tharollo ea ente Neurorubin e sebelisoa bakeng sa ente ea methapo ea kutlo; liente li khothaletsoa sethaleng se kaholimo sa mesifa ea gluteal.
Litekanyetso tsa lithethefatsi le khafetsa ea liente li latela botebo ba hypovitaminosis.
Maemong a matla, 3 ml ea lithethefatsi hangata e tsamaisoa letsatsi le leng le le leng kapa ka nako e le ngoe ka matsatsi a 2 ho fihlela tekanyo ea methapo ea bohloko e fokotseha, kamora moo ba fetohelang 3 ml ea moriana makhetlo a 1-2 ka matsatsi a 7.
Maemong a boima bo leka-lekaneng, 3 ml ea lithethefatsi hangata e tsamaisoa makhetlo a 1-2 ka matsatsi a 7.
Nako ea phekolo ea botsoali le Neurorubin e itšetlehile ka sesosa sa hypovitaminosis. Ha u etsa kalafo ea lithethefatsi ea nako e telele, li-paramente tsa laboratori li lokela ho betoa leihlo likhoeli tse ling le tse ling tse 6.

Litlamorao:
Ha o sebelisa lithethefatsi ho bakuli, ho ile ha hlokomeloa litlamorao tse latelang:
Ho tsoa ho tsamaiso ea tšilo ea lijo: ho nyekeloa ke pelo, ho hlatsa, ho eketseha ha lipilisi tsa hepatic maling. Ho bakuli ba nang le kutloisiso e eketsehileng ea motho ka mong, ho tsoa mali ho ile ha hlokomeleha ha ho nooa moriana.
Ho tloha tsamaisong ea methapo ea methapo e bohareng le e poteletseng: bofokoli, hlooho ea hlooho, ho tsekela. Maemong a ikhethileng, ho tšoenyeha, ho teneha ho eketsehileng le ho tšoenyeha ho ile ha hlokomeloa. Ha ba sebelisa lithethefatsi ka tekanyetso e phahameng, bakuli ba bang ba hlokometse ketsahalo ea "peripheral sensory neuropathy" e hlahang kamora ho khaotsa lithethefatsi.

Ho tsoa ho tsamaiso ea pelo: tachycardia, ho putlama ha mali (ho bonoang feela ho bakuli ba nang le kutloisiso e eketsehileng ea motho ka mong).
Mekhoa ea ho kulisa: ho hlohlona ha letlalo, lekhopho, urticaria, ha u sebelisa litekanyetso tse phahameng tsa moriana ho bakuli, nts'etsopele ea makhopho e ile ea lemohuoa.
Litla-morao tse ling: cyanosis, edema ea pulmonary, mofufutso. Ho bakuli ba nang le hypersensitivity ho likarolo tsa moriana, ho ka hlaha maikutlo a anaphylactoid, ho kenyeletsa edema ea Quincke. Ka tsamaiso ea batsoali ea lithethefatsi ho bakuli ba nang le hypersensitivity ho livithamini tsa B, ho ka ba le tšohanyetso ea tšohanyetso.

Contraindication:
Ho eketsa kutloisiso ea motho ka mong likarolo tsa moriana.
E laetsoe ka hloko ho bakuli ba nang le psoriasis, hobane cyanocobalamin e ka tsosa ho senyeha ho psoriasis.
Neurorubin ea lithethefatsi ka mokhoa oa tharollo ea ente ha e sebelisoe nakong ea bokhachane le pelehi, hammoho le kalafo ea bana ba ka tlase ho lilemo tse 16.

Boimana
Setlhare se tšela mekoallo ea hematoplacental 'me se ikemiselitse ho lebese la matsoele. Ha ho na datha mabapi le polokeho ea moriana nakong ea kemolo le ho lactation. Lithethefatsi nakong ea kemolo li ka laeloa ke ngaka e tlang haeba phaello e lebelletsoeng ho mme e feta kotsi e ka bang teng ho lesea. Haeba ho hlokahala ho fana ka moriana nakong ea lebone, hoa hlokahala ho etsa qeto ea ho khaotsa ho anyesa.

Ho sebelisana le lithethefatsi tse ling:
Ka tšebeliso e le 'ngoe, sethethefatsi sena se fokotsa phello ea kalafo ea levodopa, e lokelang ho tsotelloa ha u phekola bakuli ba nang le lefu la Parkinson le ho qoba tšebeliso e tšoanang ea meriana ena.
Ka tšebeliso e tšoanang, Neurorubin ea lithethefatsi e ntlafatsa chefo ea isoniazid.
Neurorubin ka lebaka la vithamine ea eona ea B6 e khona ho fokotsa katleho ea altretamine ka tšebeliso e tšoanang.
Thiosemicarbazone le fluorouracil ke bahanyetsi ba vithamine B1.
Lithethefatsi tse nang le envelop le thepa ea antacid li fokotsa ho amoheloa ha lithethefatsi Neurorubin-Forte Lactab.

Bongata
Ka tšebeliso ea lithethefatsi tse ngata ho bakuli, keketseho ea ho teba ha litlamorao e bonoa.
Ha ho na litlhare tse tobileng. Haeba ho na le overdose, gastric lavage le tsamaiso ea li-enterosorbents li bontšoa. Phekolo ke letšoao. Ka nts'etsopele ea anaphylactic makala, li-glucocorticosteroids bakeng sa ts'ebeliso ea systemic le li-antihistamines li sebelisoa.

Foromo ea tokollo:
Litafole, koaetsoe ka filimi, likotoana tse 10 ka blister, 2 lithutsoana ka lebokoseng la karete.
Tharollo ea ente ea 3 ml ka ampoule, ampoules tse 5 ka lebokoseng la karete.

Maemo a polokelo:
Setlhare se khothalletsoa hore se bolokoe sebakeng se omileng hole le khanya ea letsatsi. Matlapa a Neurorubin-Forte Lactab a khothalletsoa hore a bolokoe ka mocheso oa likhato tse 15 ho isa ho 25 tsa Celsius.
Tharollo ea ente Neurorubin e khothalletsoa hore e bolokoe ka mocheso oa likhato tse 2 ho isa ho tse 8 tsa Celsius.
Bophelo ba sehatsetsing sa moriana ka mokhoa oa tharollo ea ente ke lilemo tse 3.
Bophelo ba sehatsetsing ba lithethefatsi ka mokhoa oa matlapa ke lilemo tse 4.

Synonyms:
Neurovitan, Milgamma.

Moetso:
3 ml (1 ampoule) ea ente e na:
Thiamine hydrochloride - 100 mg,
Pyridoxine hydrochloride - 100 mg,
Cyanocobalamin - 1 mg.
Bahlomphehi.

Letlapa le 1 le koahetsoeng ka filimi le na le:
Thiamine mononitrate - 200 mg,
Pyridoxine hydrochloride - 50 mg,
Cyanocobalamin - 1 mg.
Bahlomphehi.

Hlokomela!
Pele o sebelisa lithethefatsi Neurorubin o lokela ho bona ngaka. Buka ena e fanoa phetolelong ea mahala ebile e etselitsoe merero ea tlhahisoleseling feela. Bakeng sa tlhaiso-leseling e batsi, ka kopo sheba litlhaloso tsa moetsi.
Mohloli oa litlatsetso, litaelo tsa tšebeliso ea lithethefatsi (litlhare): Setsi "Piluli - Medicine ho tloha A ho Z"

Ho batla ka boiketsetso litheko tse ntle ka ho fetisisa tsa lithethefatsi le li-analog tsa generic ho NEURORUBINE FORTE LACTAB N20 tlanya mona:


• Litšoantšo li etselitsoe litšoantšo feela. Litšoantšo tsa lithethefatsi sebakeng sa marang-rang li ka fapana ka sebopeho sa 'nete.

Ketso ea pharmacological

Moriana o na le livithamini tse tharo tse tlatselletsang le ho ntlafatsa ketso ea e mong.

Vithamine B1, kapa thiamine, e kenella phetohong ea redox ea 'mele e le coenzyme. E sebelisa lihlahisoa tsa metabolic tse nang le chefo tlas'a-oxidized - li-pyruvic le lactic acid. E laola carbohydrate, mafura le protheine metabolism.

Thiamine e khothalletsa tlhahiso ea tšusumetso haufi le methapo ea kutlo, e ntlafatsa metabolism ea methapo. E laola motility oa mala le tsamaiso ea tšilo ea lijo. E na le phello e bonolo ea analgesic maemong a phahameng.

Ka lebaka la ho haella ha vithamine B1, methapo ea kutlo e amehang (polyneuritis), kutloelo-bohloko, lefu la Wernicke-Korsakov (le nang le joala) ha le matla.

Vitamin B6, pyridoxine - ntho e kenyelitsoeng ho protheine le mafura a metaboliki, lits'ebetso tsa matla tsa lisele tsa methapo. Ke coenzyme ea phetisetso ea li-amino acid tse bokong. E khothaletsa motsoako oa li-neurotransmitter tsa bohlokoa ka ho fetisisa tsa tsamaiso ea methapo ea methapo le methapo: adrenaline, norepinephrine, dopamine. E ntlafatsa boemo ba sebete, e fokotsa lipontšo tsa lefu la matsoele a basali: ho tšoaroa ke hlooho, ho ruruha le ho mpefala ha maikutlo. E nka karolo mofuteng oa hemoglobin.

Ka lebaka la khaello ea vithamine ea B6, mokhathala, ho ruruha, ho eketseha ha prolactin ea lihormone, ho kuta moriri, ho hlohlona ha khoeli, le dermatitis ho ka hlaha.

Vitamin B12, cyanocobalamin - motsoako oa lik'hemik'hale o nang le tšepe ea cobalt. E ama protheine, metabolism ea mafura. E khothaletsa karohano ea lisele ka ho laola ho hlophisoa ha li-anemic acid. Eketsa palo ea lisele tse khubelu tsa mali maling, a nka karolo karohanong ea tsona ka lebaka la methapo ea methapo. E fokotsa cholesterol ea mali, homocysteine. Tšusumetso e ntle lits'ebetsong tsa methapo ea methapo e bohareng le e poteletseng. E khothalletsa boitšoaro bo tloaelehileng ba tšusumetso ea bohloko haufi le likhoele tsa axonal.

Ka lebaka la khaello ea vithamine B12, ho ka ba le likhathatso tse matla ts'ebetsong ea lesapo la mokokotlo, phallo ea mali e matla.

Ka lebaka la khaello ea vithamine B12, mafura a sebete a sebete a ka hlaha.

Mofumahali

Ha e nkoa ka molomo, thiamine e kenella ka mpeng e nyane ebe e kena ka har'a sebete. E 'ngoe ea eona e qaptjoa hangata. E tšelisitsoe mme e hlahisoa ka mokhoa oa thiamincarboxylic acid, dimethylaminopyrimidine. Palo e nyane ha e sa fetoloe ka moroto.

Pyridoxine hydrochloride, ha e nkuoa ka molomo, e kenella ka mafolofolo mme e kena ka har'a sebete. E etselitsoe pyridoxalphosphate le pyridoxamine. E tlama le liprotheine tse tsamaisang mali 'me li bokellana mesifa ka tsela ea pyridoxalphosphate. E pepisoa ka mokhoa oa pyridoxic acid.

Cyanocobalamin e ananeloa ke 'mele ka lebaka la kananelo e kenelletseng ea Castle e fumanoang ka mpeng - gastromucoprotein. E kenella ka mpeng, e tlameletsoe maling le liprotheine tse tsamaisang - transcobalamin le alpha-1-globulin. E bokellana sebeteng, moo e ka bolokoang nako e ka etsang selemo. Bophelo ba halofo ea mali ke matsatsi a 5.

Phekolo ea ka mpeng

Ho nyekeloa ke pelo, ho hlatsa, ho otla ha pelo, bohloko ba ka mpeng.

Sebelisa botsofaling

E amoheloa hore e sebelisoe ha e laetsoe ke ngaka mme e nahanela litlolo tsohle. Cyanocobalamin e eketsa viscosity ea mali, ka hona e ka eketsa kotsi ea thrombosis.

Cyanocobalamin e eketsa viscosity ea mali, ka hona e ka eketsa kotsi ea thrombosis.

Ho sebelisana le lithethefatsi tse ling

Li-antacid le baloi li fokotsa ho monya lithethefatsi. 6-fluorouracil, thiosemicarbazone - bahanyetsi ba thiamine.

Vitamin B6 e fokotsa mosebetsi oa lithethefatsi tse khahlanong le Parkinsonia Levodopa.

Vitamin B6 e fokotsa mosebetsi oa lithethefatsi tse khahlanong le Parkinsonia Levodopa.

Litlhahlobo tsa Neurorubin Fort

Igor ea lilemo li 40 Samara

Ke rekile livithamini bakeng sa kalafo ea osteochondrosis. Ho bile le bohloko molaleng.Kamora ho sebelisa moriana, ba ile ba fokola. O ile a qala ho ikutloa a thabile le ho feta. Mofoka o ile oa feta hoseng.

Anna, ea lilemo li 36, Kazan

Boima ba maoto le menoana e ne e tšoenyehile. Ngaka ea neuropathologist e laetse litlhare tsena. Matšoao a kokobela. Kamora ho nka matlapa, ho bile le ts'abo e nyane, litla-morao li bontšoa ka litaelo. Ho bile le hlooho e bohloko.

Contraindication

Hypersensitivity ho lithethefatsi.

Vitamin B 1 E tšoaelitsoe hore e sebelisoe mafu a kulang.

Vitamin B 6 e tšoaetsanoa haeba ho na le bothata ba peptic ulcer le mpa ea duodenum sethaleng (kaha ho ka ba le ho eketseha ha acidity ea lero la gastric).

Vitamin B 12 E tšoaetsitsoe hore e sebelisoe ho erythremia, erythrocytosis, thromboembolism.

Litšireletso tse loketseng tsa tšebeliso

Ka lebaka la hypersensitivity ho livithamini B 1 , Ho 6 B 12 nakong ea kalafo, methapo e tsoang letlalong le linama tse sa sebetseng hantle e ka hlaha.

Pyridoxine e ka tsosa ho hlaha hoa makhopho a letlalo la makhopho kapa makhopho a letlalo kapa ea ntlafatsa lipontšo tsa tse teng.

Ka kenyelletso ea vithamine 12 setšoantšo sa tliliniki, hammoho le liteko tsa laboratori bakeng sa myelosis e thabisang kapa khaello ea mali e matla, li ka felloa ke ho hlaka.

Ho nwa joala le tee e ntšo ho fokotsa ho monya ha thiamine.

Ho nwa lino tse nang le libido tsa sulphite (joalo ka veine) ho eketsa ho senyeha hoa thiamine.

Hobane moriana o na le vithamine 6 e lokela ho sebelisoa ka hloko ho bakuli ba nang le nalane ea bohloko ba ka mpeng le ea duodenal, e hlahisoang ke ho fokola ha renal le hepatic function.

Bakuli ba nang le neoplasms, ntle le linyeoe tse tsamaeang le khaello ea methapo ea methapo ea mali le khaello ea vithamine B 12 ha ea lokela ho sebelisa lithethefatsi.

Setlhare sena se sebelisoa bakeng sa ho bola ka matla kapa ka matla ho bola hoa pelo le ts'ebetso ea angina pectoris.

Sebelisa nakong ea bokhachane le pelehi

Moriana o fuoa feela kamora tlhahlobo e felletseng ea kamohelo / kotsi ea kotsi, hobane ha ho na datha e lekaneng bakeng sa polokeho ea moriana nakong ea kemolo.

Vithamine B 1 , Ho 6 B 12 e pepesitsoe lebeseng la matsoele. Litekanyetso tse phahameng tsa Vitamin B 6 e ka thibela tlhahiso ea lebese. Boithuto mabapi le secretion ea livithamini ho lebese la matsoele ha lia etsoa. Qeto ea ho emisa ho anyesa kapa ho sebelisa sethethefatsi e tlameha ho etsoa ho nahanela bohlokoa ba ho sebelisa meriana bakeng sa mme. Haeba ho hlokahala, ts'ebeliso ea lithethefatsi e lokela ho emisa ho anyesa nakong ena.

Bokhoni ba ho susumetsa sekhahla sa karabelo ha ho khanna likoloi kapa mekhoa e meng

Setlhare ha se ame bokhoni ba ho khanna makoloi kapa ho sebetsa ka methapo.

Maemong moo ho tsekela ho ella hloko nakong ea ts'ubuhlellano ea mahlo nakong ea kalafo, motho o lokela ho hana ho khanna makoloi le ho sebetsa ka methapo.

Bana ha baa lokela ho fuoa moriana, hobane ha ho na boiphihlelo ka tšebeliso ea bana.

Bongata

Vitamin B 1 : e na le mefuta e mengata ea kalafo. Methapo e phahameng haholo (e fetang 10 g) e bonts'a phello ea mokokotlo, e hatelletseng ts'usumetso ea methapo ea methapo.

Vitamin B 6 : E na le chefo e tlase haholo. Tšebeliso ea nako e telele (ho feta likhoeli tse 6-12) ka tekanyetso ea vithamine B e fetang 50 6 letsatsi le leng le le leng li ka lebisa ho peripheral sensory neuropathy.

Ts'ebeliso e Ntle ea Vitamin 6 litekanyetso tse fetang 1 g ka letsatsi ka likhoeli tse 'maloa li ka lebisa litlamorao tsa neurotoxic.

Li-neuropathies tse nang le mathata a ho ferekana le kutloelo-bohloko, ho ts'oaroa ha methapo ea kutlo le liphetoho ho EEG, hammoho le maemong a mang hypochromic anemia le seborrheic dermatitis li ile tsa hlalosoa kamora ho tsamaisoa ha ≥ 2 g ka letsatsi.

Vitamin B 12 : kamora ho tsamaisoa ke batsoali (maemong a sa tloaelehang, ka mor'a taolo ea molomo), lintho tse kulang, mathata a letlalo le eczematous le mofuta o mosesaane oa makhopho li ile tsa bonoa ho litekanyetso tse phahameng ho feta tse khothalelitsoeng.

Ka tšebeliso ea nako e telele litekanyetso tse phahameng, tlolo ea ts'ebetso ea li-enzyme tsa sebete, bohloko pelong, le hypercoagulation lia khonahala.

Phekolo ea ho ts'oara joala ka hanong: ho felisoa ha ntho e chefo (ho hlatsa, hlatsoa mpa), mehato ea ho fokotsa ho amoha (ts'ebeliso ea mashala a entsoeng ka letsoho).

Litlamorao

Ho tsoa ho sesole sa 'mele: hypersensitivity reaction, anaphylactic shock, anaphylactic shock. Litla-morao tse ke keng tsa etsahala.

Ho tsoa tsamaisong ea endocrine: Ho hlahisoa ha prolactin hoa thibeloa.

Ho tsoa tsamaisong ea methapo: ho tšoenyeha, tšebeliso ea nako e telele (ho feta likhoeli tse 6-12) tsa vithamine 6 ka tekanyetso ea ≥ 50 mg letsatsi le letsatsi, e ka lebisa ho pherekano ea methapo ea kutlo, ho ruruha ha methapo, malaise, ho tsekela, hlooho.

Ho tsoa ho tsamaiso ea pelo le pelo: tachycardia, ho oa.

Karolong ea mokhoa oa ho hema, sefuba le mediastinum: cyanosis, pulmonary edema.

Ho tsoa pampiring ea ka mpeng: mathata a ka mpeng, ho kenyelletsa ho nyekeloa, ho hlatsa, lets'ollo, bohloko ba ka mpeng, ho eketsa acidity ea lero la gastric.

Ho tsoa ho sebete le senya. ha e sebelisoa ka tekanyetso e phahameng, keketseho ea boemo ba glutamic acid-transmucosal transaminase (SGOT) serum.

Ka lehlakoreng la letlalo le lisele tse nyane: lekhopho, mokokotlo oa letlalo, ho kenyeletsa pruritus, urticaria.

Mathata a mang: ho fufuleloa ho feteletseng, maikutlo a bofokoli, ho tsekela, ho holofala.

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